GABASIGN 800 CAP is a high-potency formulation containing Gabapentin 800 mg, developed to provide effective relief from chronic neuropathic pain and as an adjunctive therapy in the treatment of partial-onset seizures. Gabapentin is a structural analogue of GABA (gamma-aminobutyric acid) that modulates calcium channels in the nervous system to reduce nerve excitability and pain signaling.
This advanced pharmaceutical product is manufactured by BluepillExpress, a leading Indian third-party manufacturing company globally recognized for quality, regulatory excellence, and consistent supply chain execution. Each capsule is manufactured using advanced machinery and under rigorous quality control to meet global export requirements across regulated and semi-regulated markets.
Indications
Diabetic peripheral neuropathy
Postherpetic neuralgia
Partial seizures (adjunct therapy)
Fibromyalgia (off-label use)
Central pain syndrome
Nerve pain from spinal cord injuries or shingles
Mechanism of Action
Gabapentin acts by binding to the α2δ subunit of voltage-gated calcium channels in neurons, inhibiting the release of excitatory neurotransmitters such as glutamate, substance P, and norepinephrine. This helps reduce abnormal nerve firing and relieves neuropathic pain and seizures.
Dosage & Administration
Typical Dose Range: 300–3600 mg/day
GABASIGN 800 CAP is used in patients titrated to higher daily doses for stable long-term management
Dose to be taken as prescribed by a physician; often administered 2-3 times per day
Must not be stopped abruptly; gradual tapering is advised
Pharmacokinetics
Absorption: Dose-dependent (bioavailability decreases with increasing dose)
Tmax: 2–3 hours post-administration
Half-life: 5–7 hours
Elimination: Renal (unchanged)
Metabolism: Not significantly metabolized in the liver
Advantages of GABASIGN 800 CAP
High-dose capsule provides enhanced control of neuropathic symptoms
Non-sedative and non-addictive alternative to opioids
Suitable for patients who require less frequent dosing due to sustained concentration
Manufactured under GMP-certified facilities with complete quality assurance
Available for custom branding, bulk supply, and private labeling
Description provided by bluepill express.
FIEO Registered
Export Ready
